Idebenone
antioxidant health benefit and research studies
Idebenone is a synthetic analogue of coenzyme Q10 used in Europe in the
treatment of vascular and degenerative diseases of the central nervous system.
Idebenone is a strong antioxidant
and gaining popularity.
Alzheimer's disease treatment
Studies with
Idebenone in regards to therapy of
Alzheimer's
disease have been inconsistent, but there may be a trend for a slight benefit.
Idebenone treatment fails to slow
cognitive decline in Alzheimer's disease.
Neurology. 2003. Department of
Neurosciences, University of California San Diego School of Medicine, La Jolla, USA.
To determine the effect of idebenone on the rate of decline in Alzheimer's
disease. A 1-year, multicenter, double-blind, placebo-controlled, randomized
trial was conducted. Subjects were over age 50 with a diagnosis of probable AD
and had Mini-Mental State Examination (MMSE) scores between 12 and 25. Subjects
were treated with idebenone 120, 240, or 360 mg tid, each of which was compared
with placebo. Idebenone failed to slow cognitive decline in AD that was of
sufficient magnitude to be clinically significant.
Friedreich's ataxia treatment
Idebenone may be helpful in Friedreich's ataxia.
Neurological effects of high-dose
idebenone in patients with Friedreich's ataxia: a randomised, placebo-controlled
trial.
Lancet Neurol. 2007.
Friedreich's ataxia
is a progressive, multisystem, degenerative disorder caused by a reduction in
frataxin. Loss of frataxin results in mitochondrial dysfunction and oxidative
damage in patients and model systems. Previous studies have indicated that the
antioxidant idebenone (5 mg/kg daily) reduces cardiac hypertrophy, but definite
improvement in neurological function has not been shown. 48 genetically
confirmed Friedreich's ataxia patients, aged 9-17 years, were enrolled in a
6-month, randomised, double-blind, placebo-controlled study. The patients
received placebo or one of three doses of idebenone (approximately 5 mg/kg, 15
mg/kg, and 45 mg/kg), stratified by body weight. Treatment with higher doses of
idebenone was generally well tolerated and associated with improvement in
neurological function and ADL in patients with Friedreich's ataxia. The degree
of improvement correlated with the dose of idebenone, suggesting that higher
doses may be necessary to have a beneficial effect on neurological function.
Idebenone treatment in Friedreich patients: one-year-long randomized
placebo-controlled trial.
Neurology. 2003.
The authors carried out a 1-year, randomized, placebo-controlled trial of
idebenone in 29 patients with Friedreich ataxia. They found significant
reductions of interventricular septal thickness and left ventricular mass in the
idebenone group vs the placebo group, with no improvement in other heart
ultrasound measures or neurologic condition. The absolute cardiac changes were
modest, but the findings suggest that larger trials should assess whether
idebenone reduces ventricular hypertrophy in patients with Friedreich ataxia.
Huntington's
disease
Idebenone has not been found to be helpful
in Huntington's disease.
Idebenone side effects,
safety
The most common side effects associated with idebenone are
insomnia, stomach
pain, nausea, and anxiety.